Inside story of the drug Carisoprodol

Carisoprodol is identified under the generic brand name Soma. It is a prescription-based medicine mainly used for treating numerous human muscular-skeletal disorders. Soma 350 mg is highly used among adults to treat muscle spasms or injuries. Also, it is one of the well-known anti-depressant brands that works centrally by developing the soothing effect with less potential for addiction. With the convenience of an online pharmacy, you may buy Pain O Soma 350 mg with free US-US shipping and for other international shipping, you may avail of multiple discount alerts on all your medicinal products using verified online pharmacists.

History of Carisoprodol

The inside story of the drug Carisoprodol was narrated by a group of pharmacologists in the United States. On 1st June, numerous American pharmacists from different states were gathered at a University located at Wayne State in Detroit, Michigan, in the year 1959. The gathering was scheduled to talk over a new drug that would contain sterile and muscle relaxant properties.

After a healthy discussion, Mr. Frank Berger came with an antiseptic drug named Carisoprodol developed at Wallace Laboratories.

The origin of this drug is derived from the existing metabolite known as meprobamate. It withholds the sedative substances along with a barbiturate effect. The extent of these substances is added more safely and efficiently to treat the syndrome.

Carisoprodol is a muscle relaxant with less potential for dependence and addiction if consumed in an adequate proportion for the acute duration.

It is also known by the brand name Soma or Rela, which is formed as a safer and efficient version of meprobamate.

Medical genuine uses

FDA duly approves carisoprodol for genuine medical uses related to the human skeletal disorder. Many people suffering from back, neck, or spinal pain find it difficult to concentrate at work or school. Sometimes, their pain also shifts from acute to chronic condition, making it tough to fulfill daily household chores and restricted mobility.

In such cases, this drug acts as a discomfort relieving agent related to painful muscular disorders. As carisoprodol is marketed with the brand name Soma available from 350 mg onwards is mainly used as a muscle relaxant. Along with its spasms relaxing properties, it also exhibits a soothing effect by relaxing the painful sensations entering the peripheral nervous system.

Many physicians prescribe this medication for those suffering from anxiety and tension, as it releases tranquilizing effects present in the parent compound belonging to the benzodiazepine class of drugs.

It is also indicated to help with muscle spasms, spasticity, injuries, sprains, strains, and inflammation by relaxing the affected area.

Apart from this, health-care practitioners also consider it as a suitable drug for myofascial syndrome along with proper rest and alternative physical therapy for better results.

Mechanism of action of a Schedule Drug

Carisoprodol performs centrally by relaxing the muscle spasms indirectly by calming the pain outrage travelling from the nerves to the nervous system. Its parent agent is classified under schedule substance IV in 1970 due to its narcotic effect and marketed under several brand names such as Pain O Soma, Carisoma, Prosoma, and many others.

The primary meprobamate is responsible for altering the painful sensations in the interneuron activity in the spinal region by forming a descending network in the brain. This metabolite is also in charge of spreading the therapeutic effect by making a person feel relaxed by creating a wall against painful signals.

However, meprobamate may turn into an abusive agent if overdosed. Therefore, it is highly recommended to consult your doctor regarding the dose regimen and do not use this medication for a prolonged duration.

Medical administration

The suitable dose of Soma hybrid is one to two tablets four times a day, applicable for adults. A single pill is composed of a mixture of Carisoprodol 350 mg.

Although it is an active muscle relaxant, it is not suitable for children below 16 years of age and older people above 65 years of age due to its sedative effect.

The maximum daily measure of Soma should not be more than 1600 mg, and the weekly prescription should not be exceeding up to two to three weeks.

It is available under the generic brand known as Soma 350 mg, which you may have with or without a meal as per your doctors’ advice and if you do not have gastrointestinal problems.

As per the blister instructions, you may have Pain O Soma 350 mg along with proper rest and diet and physical therapy such as yoga or exercise for adequate recovery.

How is it supplied and stored?

Carisoma 350 mg tablet comes in a two-layered white, circular-shaped, engraved with SOMA on the saffron layer with 37 WALLACE 2001 belongs to a tranquilizer and muscle relaxant class of drugs.

For storage, you may store the bottle at a room temperature of 68-to-77-degree F; also, make sure to protect it from moisture and keep your container tightly locked after every use.

Abuse of the drugs

Carisoprodol contains an active compound known as meprobamate, which belongs to the abusive class of drugs. But FDA has scheduled it under the tranquilizing medications category due to its muscle calming properties.

Although, many abusive cases have been suspected after its post–marketing survey. The primary reason for its abuse was due to prolonged consumption.

Another cause of dependence was due to the patient’s previous addiction, medical history, or other combination of drugs.

To decrease the prospect of abuse or dependency, one should take carisoprodol with care and with health-care expert’s advice.

For those taking other anti-depressants should not take Soma for more than 2 – 3 weeks of duration. As primarily acute pain is resolved or treated within two weeks.

Also, abrupt stoppage should be avoided after chronic use as it may lead to withdrawal symptoms.

Side-effects

Carisoprodol Side Effects

The common adverse effects have been administered post-FDA approval for the use of Soma medication. This reaction occurs after the interaction of drug with the human system:

  • Effect on central nervous system: Drowsiness, vertigo, head pain, tremor, anxiety, tension, frustration, seizures, and insomnia.
  • Effect on the cardiorespiratory system: Postural hypotension, irregular breathing, respiratory depression, facial redness, or flushing.
  • Effect on the gastrointestinal system: Vomiting, stomach pain, nausea, hematologic, leukocytosis, and diarrhea.

The above adverse effects can affect both physically and psychologically; therefore, alerting exercise such as driving or riding should be avoided for life safety. Also, overdose or prolonged use should not be done to prevent effects on the peripheral nervous system.

However, if you are experiencing severe sedation sensations, quickly seek professional help to prevent further fatal issues.

Over-dose

Overdose of Soma develops depression, respiratory depression, hypotension, delirium, hallucinations, blurred eyesight, euphoria, restricted mobility, brain tumor, coma, or even death.

A few cases of CNS problems have been reported after an excess dose of Carisoprodol. This overdose mainly occurs due to consuming multiple anti-depressants simultaneously or consuming Soma without prescription and alcohol.

It is highly advisable to make ethical use of this medicinal drug and always follow the guidelines given by your physician and read the generic information provided on the label to be aware of the pros and cons of the medicine.

References

Anon, 1997. Carisoprodol. Environmental Health Perspectives, 105, p.283. Available at: http://dx.doi.org/10.2307/3433446.

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