Metaxalone (Skelaxin) is the prescribed muscle relaxant medication for treating musculoskeletal pain and discomfort. It was first approved by the U.S. Food and Drug Administration (FDA) in 1962. The drug was originally developed by the pharmaceutical Company Wallace Laboratories, later acquired by Carter-Wallace.
A Short Brief Of Metaxalone
Skelaxin is the brand name of Metaxolone. It is used to treat muscle pain and discomfort caused by musculoskeletal conditions, such as strains, sprains, or other injuries.
Metaxalone is a prescription medication and should only be used under the guidance of a healthcare professional. It is important to follow the dosage instructions provided by your doctor and to report any side effects of concern to them.
Metaxalone is most likely a narcotic since it is an opioid, which can provide morphine-like effects to relieve pain and is possibly addictive.
How Does Metaxalone Work?
The exact mechanism of Metaxalone is not fully understood yet. It is thought that Metaxalone works by blocking the pain sensation transmission between the nerves and the central nervous system.
Metaxalone works by increasing the activity of the neurotransmitter called gamma-aminobutyric acid (GABA), which helps reduce nerve cells in the brain and spinal cord that control muscle movement. By enhancing GABA activity, Skelaxin can help decrease muscle pain and discomfort.
Usages Of Metaxalone
As mentioned above, Metaxalone, an active ingredient in Skelaxin, is a muscle relaxant used to treat muscle spasms caused by musculoskeletal conditions such as strains, sprains, or other injuries.
Dosages, Forms And Strengths Of Metaxalone
Adults typically take 800 mg three or four times a day.
For youngsters aged 13 to 18, the exact dosage of 800 mg administered three to four times per day is used.
Children under the age of 12 should not be administered this medication.
Take the missed dose immediately if it will be a while until your next dosage. To protect the missing dosage, never combine two doses. Taking two doses at once might have greater harmful impact on your health.
Seek emergency medical attention if you take too much Metaxalone since it might have harmful effects. Due to the significant sleepiness it may produce, it may also be lethal.
Who shouldn't take it, exactly?
Metaxalone should not be taken:
- Under 12 Years Old
- Allergic to Metaxalone
- liver and kidney disease
- regular alcohol consumption
- a blood condition
- MAO inhibitor is taken two weeks earlier
Pregnant and breastfeeding women should not take Metaxalone as it can affect the health of both women and the child. The doctor can only prescribe it in necessary extreme conditions.
Forms and Strengths
- Metaxalone comes in tablet form.
- Strengths of Metaxalone are 400mg, 640mg, and 800mg
Precautions To Be Taken For Metaxalone
Metaxalone (Skelaxin) is a prescription medication that should only be taken with the proper precautions.
Here are some precautions for Metaxalone:
- Inform your doctor about the medical health conditions you have, including kidney or liver disease, anemia, or allergies
- Inform your doctor about the medication you are using before taking Metaxalone, including over-the-counter medicines and supplements.
- Follow the dosing instruction prescribed by your doctor, and do not overdose on the Metaxalone. It may cause side effects.
- Avoid driving or operating heavy machinery, which needs alertness.
- If you are facing any side effects, such as an allergic reaction, rash, sink allergies, or difficulty in breathing, immediately stop taking it and visit the doctor
- Store metaxalone at room temperature and keep it away from direct sunlight.
- Use Metaxalone (Skelaxin) according to the prescription and follow the precaution properly to avoid the Skelaxin side effects.
Side Effects Of Metaxalone
Metaxalone (Skelaxin) can cause a range of side effects which vary from person to person: here are the table of common side effects and serious side effects of Metaxalone (Skelaxin).
Common side effects
Serious side effects
Note that this table is not comprehensive, and other side effects may be associated with metaxalone. It is important to talk to your healthcare professional if you experience any side effects while taking metaxalone, especially if they are severe or persistent.
Interactions Of Metaxalone
Metaxalone (Skelaxin) may interact with other medications and substances, which may affect the effectiveness of the Metaxalone and may cause serious side effects.
Central nervous depressant: taking Metaxalone with other medication that depresses the central nervous system, such as opioids, benzodiazepines, or alcohol, can increase the risk of drowsiness, dizziness, and difficulty breathing. Metaxalone will make you sleepy because all muscle relaxers have this effect.
CYP3A4 inhibitor: medication that inhibits the CYP3A4 substance, such as erythromycin, ketoconazole, and grape juice, can enhance the effects of metaxalone in the body, which can increase the risk of side effects.
Warfarin: Metaxalone can enhance the anticoagulant effect of warfarin, which can raise the risk of bleeding
Antihistamines: taking Metaxalone with antihistamines such as diphenhydramine and chlorpheniramine can increase the risk of dizziness and drowsiness
Muscle relaxant: Taking Metaxalone with Baclofen or cyclobenzaprine, or another muscle relaxant may increase the risk of side effects.
Can You Buy Metaxalone Online?
Yes, you can buy Metaxalone (Shelaxin) online, but a prescription from a certified doctor is mandatory to buy Flexeril online from a legal pharmacy.
Before buying Metaxalone online, make sure to choose a reputable and certified pharmacy. Look for a pharmacy website that is approved by FDA and displays the FDA seal on its site. Which indicates that they are licensed and operate in compliance with state and federal laws.
There are many fraudulent websites that sell counterfeit or substandard medication. So be aware of fake and illegal pharmacies while buying metaxalone online.
Can You Buy Metaxalone Over The Counter?
No, Metaxaloine is a prescription medication it is unavailable over the counter. You need a valid prescription from a licensed healthcare provider to purchase Metaxalone.
Buying Metaxalone over the counter without a prescription is an illegal act.
As mentioned above, Metaxalone is the muscle relaxant medication used to treat musculoskeletal pain and discomfort. Although it is not a controlled substance it has the potential to cause addiction and abuse. So prescription from a certified doctor is mandatory to buy Metaxalone. Use it according to the prescription and guidelines given by your doctor. Do not increase the dose or duration of the medication.